Stereoselective Synthesis of α-Amino-C-phosphinic Acids and Derivatives
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چکیده
منابع مشابه
Stereoselective Synthesis of α-Amino-C-phosphinic Acids and Derivatives.
α-Amino-C-phosphinic acids and derivatives are an important group of compounds of synthetic and medicinal interest and particular attention has been dedicated to their stereoselective synthesis in recent years. Among these, phosphinic pseudopeptides have acquired pharmacological importance in influencing physiologic and pathologic processes, primarily acting as inhibitors for proteolytic enzyme...
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Due to their potential biomedicinal and synthetic applications, b-amino acids have attracted a great deal of attention recently [1–6]. The derived b-peptides of several amino acids have been reported to exhibit certain secondary structures and special stability against peptidase [7,8]. For example, the b-oligopeptides of six b-amino acid residues form stable helices in methanol [8]. Furthermore...
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ژورنال
عنوان ژورنال: Molecules
سال: 2016
ISSN: 1420-3049
DOI: 10.3390/molecules21091141